Fingerprint Fingerprint is based on mining the text of the persons scientific documents to create an index of weighted terms, which defines the key subjects of each individual researcher.

HIV-1 Medicine & Life Sciences
HIV Integrase Inhibitors Medicine & Life Sciences
Integrases Medicine & Life Sciences
HIV Integrase Medicine & Life Sciences
Neoplasms Medicine & Life Sciences
Acids Medicine & Life Sciences
Catalytic Domain Medicine & Life Sciences
Antiviral Agents Medicine & Life Sciences

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Research Output 1990 2017

Discovery of novel 3-hydroxypicolinamides as selective inhibitors of HIV-1 integrase-LEDGF/p75 interaction

Zhang, F. H., Debnath, B., Xu, Z. L., Yang, L. M., Song, L. R., Zheng, Y. T., Neamati, N. & Long, Y. Q. 2017 In : European Journal of Medicinal Chemistry. 125, p. 1051-1063 13 p.

Research output: Contribution to journalArticle

HIV Integrase Inhibitors
Integrases
HIV-1
HIV Integrase
Dimerization

Identification and preclinical evaluation of SC144, a novel pyrroloquinoxaline derivative with broad-spectrum anticancer activity

Grande, F., Aiello, F., Garofalo, A. & Neamati, N. May 1 2016 In : Mini-Reviews in Medicinal Chemistry. 16, 8, p. 644-650 7 p.

Research output: Contribution to journalArticle

Neoplasms
Lead
Standard of Care
Tumor Cell Line
Heterografts

Mechanistic evaluation and transcriptional signature of a glutathione S-transferase omega 1 inhibitor

Ramkumar, K., Samanta, S., Kyani, A., Yang, S., Tamura, S., Ziemke, E., Stuckey, J. A., Li, S., Chinnaswamy, K., Otake, H., Debnath, B., Yarovenko, V., Sebolt-Leopold, J. S., Ljungman, M. & Neamati, N. Oct 5 2016 In : Nature Communications. 7, 13084

Research output: Contribution to journalArticle

Glutathione Transferase
Neoplasms
Drug Delivery Systems
Cytoskeleton
Drug Resistance

Targeted Nanoparticles for the Delivery of Novel Bioactive Molecules to Pancreatic Cancer Cells

Sanna, V., Nurra, S., Pala, N., Marceddu, S., Pathania, D., Neamati, N. & Sechi, M. Jun 9 2016 In : Journal of Medicinal Chemistry. 59, 11, p. 5209-5220 12 p.

Research output: Contribution to journalArticle

Pancreatic Neoplasms
Nanoparticles
Adenocarcinoma
Plectin
Quinazolinones
6 Citations

Discovery of Novel CXCR2 Inhibitors Using Ligand-Based Pharmacophore Models

Ha, H., Debnath, B., Odde, S., Bensman, T., Ho, H., Beringer, P. M. & Neamati, N. Aug 24 2015 In : Journal of Chemical Information and Modeling. 55, 8, p. 1720-1738 19 p.

Research output: Contribution to journalArticle

Ligands
Inflammation
model
Arrestin
Cell Movement